Molecular Basis for the N-Terminal Bromodomain and Extra Terminal (BET) Family Selectivity of a Dual Kinase-Bromodomain Inhibitor

Divakaran, A.; Talluri, S. K.; Ayoub, A. M.; Mishra, N.; Cui, H.; Widen, J. C.; Berndt, N.; Zhu, J.; Carlson, A. S.; Topczewski, J. J.; Schönbrunn, E.; Harki, D. A.; Pomerantz, W. C. K.  J. Med. Chem., 2018, 61, 9316–9334.